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Synthesis and electrophysiological evaluation of 6,11-dihydrodibenzo[c,f][1,2,5]thiadiazepine-5,5-dioxide (DBTD): non-competitive GABAA receptor antagonists
(2013)
"En este trabajo describimos un nuevo proceso para obtener dibenzo[c,f][1,2,5]tiadiazepinas (DBTDs o 2) y sus efectos como modulador de los receptores GABAA de neuronas mientéricas de cobayo. La síntesis de derivados de ...
Dibenzo[1,2,5]thiadiazepines are non-competitive GABAA receptor antagonists
(MDPI, 2013)
"A new process for obtaining dibenzo[c,f][1,2,5]thiadiazepines (DBTDs) and their effects on GABAA receptors of guinea pig myenteric neurons are described. Synthesis of DBTD derivatives began with two commercial aromatic ...